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Cat No. | Product Name | Synonyms | Targets |
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TP1732L | Galanin (1-30), human acetate | Galanin (1-30), human acetate(119418-04-1 Free base) | Others |
Galanin (1-30), human acetate (Galanin ) is a 30-amino acid neuropeptide. Galanin (1-30), human acetate acts as an agonist of GalR1 and GalR2 receptors, with Kis of both 1 nM. | |||
T60193 | CB-5339 | p97 | |
p97-IN-1 is a potent inhibitor of p97 with an IC 50 <30 nM [1]. | |||
T2081 | LY2409881 trihydrochloride | LY2409881 | Apoptosis , IκB/IKK |
LY2409881 trihydrochloride is a novel specific inhibitor of IKK2 (IC50: 30 nM); IC50 for IKK1 and other common kinases is at least one log higher. | |||
T25175 | BRD 9757 | BRD9757,N-Hydroxy-1-cyclopentene-1-carboxamide,BRD-9757 | HDAC |
BRD 9757 (N-Hydroxy-1-cyclopentene-1-carboxamide) is a selective inhibitor of HDAC6 (IC50 = 30 nM). | |||
T13362 | XY101 | ROR | |
XY101 is a selective, metabolically stable and orally available agonist of RORγ inverse(IC50 of 30 nM and a Kd of 380 nM). | |||
T74809 | STING agonist-30 | STING , Antifection | |
STING agonist-30 is a potent STING agonist that triggers STING-dependent immune activation.STING agonist-30 shows broad-spectrum inhibitory effects against a variety of viruses including HSV (Herpes Simplex Virus), rotav... | |||
T5099 | Gefapixant | RO 4926219,AF219,MK-7264 | P2X Receptor |
Gefapixant (AF219) is a P2X3 receptor (P2X3R) antagonist with IC50 of ~30 nM at recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. | |||
T76089 | Pepinh-TRIF TFA | Raf , TLR | |
Pepinh-TRIF TFA is a 30 aa peptide associated with the immune system that blocks TRIF signaling by interfering with TLR-TRIF interaction (TLR-TRIF interaction ). | |||
TP2498 | Tetrapeptide-30 Acetate | Tetrapeptide-30 Acetate(1036207-61-0 Free base) | Others |
Tetrapeptide-30 Acetate (Tetrapeptide-30 Acetate) is a synthetic peptide containing the amino acids proline, glutamic acid, and lysine. It acts on and within specific targets of skin to reduce factors and interrupt the p... | |||
T10431 | Golidocitinib | AZD4205 | JAK |
Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: >14.7, >30 μM). | |||
T83966 | LSD1-IN-30 | Histone Demethylase | |
LSD1-IN-30 is a lysine-specific demethylase 1 (LSD1) inhibitor with anticancer activity for the study of small cell lung cancer and acute myeloid leukemia. | |||
T61316 | HTS07545 | NADPH | |
HTS07545 is a potent sulfide:quinone oxidoreductase inhibitor (IC50: 30 nM).HTS07545 reduces the rate of hydrogen sulfide (H2S) decomposition.HTS07545 has been used in heart failure studies. | |||
T8375 | ML-210 | CID 49766530 | Ferroptosis , GPX , Glutathione Peroxidase , Ras |
ML-210 (CID 49766530) is a selective RAS and covalent glutathione peroxidase 4 (GPX4) inhibitor(GPX4, EC50 : 30 nM), with anti-cancer activity | |||
T5403 | ULK-101 | Autophagy | |
ULK-101 is a potent and selective ULK1 inhibitor ( IC50s: 8.3/30 nM for ULK1/ULK2). It can suppress autophagy. | |||
T2414 | Torkinib | PP 242 | Apoptosis , Mitophagy , PI3K , mTOR , Autophagy |
Torkinib (PP 242) (PP 242) is a selective and ATP-competitive mTOR inhibitor (IC50: 8 nM). It also inhibits mTORC1/2 (IC50s: 30/58 nM). | |||
TP2009L | K 41498 aceate | CRFR | |
K41498 acetate, an analogues of antisauvagine-30 (aSvg-30), inhibits sauvagine-stimulated cAMP accumulation in hCRF2α- and hCRF2β-expressing cells. K41498 acetate is a potent and highly selective antagonist CRF2 receptor... | |||
T32490 | L-161240 | L-161,240 | Antibacterial |
L-161240 is an antimicrobial agent associated with lipid A biosynthesis with an IC50 value of 30 nM as determined by DEACET and a MIC value of 1-3 μg/ mL against wild-type E. coli. | |||
T6139 | A-674563 | A674563 | ERK , GSK-3 , Akt , PKA , CDK |
A-674563 is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC. | |||
T9042 | Teriflunomide impurity 3 | 4-Amino-N-(4-trifluoromethylphenyl)benzamide | COX |
Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) is a selective COX-1 inhibitor(IC50 of 30 μM). It is less active against COX-2 (IC50>100 μM). | |||
T60082 | HDAC-IN-40 | HDAC | |
HDAC-IN-40 is a potent alkoxyamide-based HDAC inhibitor with Ki of 60 nM and 30 nM for HDAC2 and HDAC6, respectively. HDAC-IN-40 had antitumor effects | |||
T9672 | GRL-0496 | SARS-CoV | |
GRL-0496 is a potent inhibitor with an enzyme inhibitory activity against SARS-CoV 3CLpro with an IC50 of 30 nM and antiviral potency with an EC50 value of 6.9 μM. | |||
T6139L | A-674563 2HCl(552325-73-2(fb-2hcl)) | ERK , Akt , PKA , CDK , PKC | |
A-674563 2HCl is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC. | |||
TQ0267 | Endomorphin 1 | Endomorphin-1 | Opioid Receptor |
Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM). | |||
T6996 | SU 5402 | SU5402 | VEGFR , FGFR , PDGFR |
SU 5402 is a potent multi-targeted receptor tyrosine kinase inhibitor with IC50 of 20 nM, 30 nM, and 510 nM for VEGFR2, FGFR1, and PDGF-Rβ, respectively. | |||
T6782L | Benzocaine xHCl(94-09-7(free base)) | Sodium Channel | |
Benzocaine shares a common receptor with all othe rLAs in the voltage-gated Na+ channel(IC50 of 0.8 mM tested with a potential of +30 mV). | |||
T29457L | 5-Hydroxydecanoate sodium | Potassium Channel | |
5-Hydroxydecanoate sodium is a selective ATP-sensitive K+ (KATP) channel blocker with IC50 of about 30 μM. 5-Hydroxydecanoate sodium is a substrate for mitochondrial outer membrane acyl-CoA synthetase with antioxidant p... | |||
T6900 | MS023 | Histone Methyltransferase | |
MS023 is a potent, selective, and cell-active Type I PRMT inhibitor with IC50 of 30 nM, 119 nM, 83 nM, 4 nM, and 5 nM for PRMT1, PRMT3, PRMT4, PRMT6 and PRMT8, respectively. | |||
T17271 | YKL-05-099 | SIK | |
YKL-05-099 is an inhibitor of the salt-inducible kinase(SIK1 and SIK3 ; IC50s: 10 and 30 nM, respectively). It has a slightly less potent SIK2-inhibitory (IC50:40 nM). | |||
T8974 | ML-211 | Others | |
ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM) | |||
T2276 | RI-1 | RI1,RAD51 inhibitor 1 | DNA/RNA Synthesis |
RI-1 (RAD51 inhibitor 1) is a RAD51 inhibitor (IC50: 5-30 μM). | |||
T72026 | P53-MDM2-IN-1 | Mdm2 , p53 | |
p53-MDM2-IN-1 (Example 30), an inhibitor targeting the p53-MDM2/X protein interaction, exhibits a K i value of 23.35 µM. This compound holds potential for applications in anti-tumor research. | |||
T9315 | 2H-Imidazo[4,5-b]pyrazin-2-one, 1,3-dihydro-6-[6-(1-hydroxy-1-methylethyl)-3-pyridinyl]-1-[(tetrahydro-2H-pyran-4-yl)methyl]- | Others | |
2H-Imidazo[4,5-b]pyrazin-2-one, 1,3-dihydro-6-[6-(1-hydroxy-1-methylethyl)-3-pyridinyl]-1-[(tetrahydro-2H-pyran-4-yl)methyl]- is a potent mTOR inhibitor with IC50 of 0.176 μM and >30 μM for mTOR and PI3Kα, respectively. | |||
T6930 | Pazopanib Hydrochloride | GW786034,Pazopanib HCl,GW786034 HCl,Votrient HCl,Armala | c-Fms , VEGFR , FGFR , PDGFR , c-Kit , Autophagy |
Pazopanib Hydrochloride (Votrient HCl) is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FGFR, c-Kit and c-Fms with IC50 of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM in cell-free assays, resp... | |||
T67887 | BDCRB | ||
BDCRB inhibits herpesvirus DNA maturation. BDCRB causes the HCMV terminase to skip the normal cleavage site and to continue to package DNA until a second cleavage site is encountered 30 kb further along the concatemer. | |||
T3073 | PF-670462 | PF670462 | Casein Kinase |
PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations. | |||
T6434 | CCG-50014 | CCG 50014 | GTPase |
CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM. | |||
T1448 | Dasatinib | BMS-354825 | Apoptosis , Bcr-Abl , Src , c-Kit , Autophagy |
Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive. Dasatinib has antitumor activity and is used in the treatment of leukemia and ly... | |||
T9711 | OGT-IN-2 | Others | |
OGT-IN-2 is a potent O-GlcNAc transferase (OGT) inhibitor. OGT-IN-2 inhibits sOGT and ncOGT with IC50 values of 30 μM and 53 μM, respectively[1]. OGT-IN-2 can be used for the research of articular diseases[1]. | |||
T27682 | CCR2 antagonist 5 | JNJ-41443532,JNJ-41443532 Free Base,JNJ 41443532,JNJ41443532 | CCR |
CCR2 antagonist 5 (JNJ-41443532) is a selective and orally active hCCR2 inhibitor with good binding affinity (IC50=37 nM) and potent functional antagonism (chemotaxis IC50=30 nM).JNJ-41443532 binds mCCR2 with a Ki of 9.6... | |||
TP1722L | PACAP (6-38), human, ovine, rat acetate | PACAP | |
PACAP (6-38), human, ovine, rat acetate is a potent PACAP receptor antagonist with IC50s of 30, 600, and 40 nM for PACAP type I receptor, PACAP type II receptor VIP1, and PACAP type II receptor VIP2, respectively. | |||
T10477 | BAY-985 | IκB/IKK | |
BAY-985 is a potent, selective, and orally active ATP-competitive dual inhibitor of TBK1 and IKKε (IC50s: 2/30 and 2 nM for TBK1 (low/high ATP) and IKKε) with antitumor efficacy. | |||
T5398 | BMS 599626 2HCl (873837-23-1(HCl)) | AC480 dihydrochloride | HER |
BMS 599626 2HCl (873837-23-1(HCl)) (AC480 dihydrochloride) is a selective inhibitor of HER1 and HER2 (IC50s: 20 nM and 30 nM), ~8-fold less potent to HER4, >100-fold to Lck, VEGFR2, c-Kit, MET, etc. | |||
T6296 | RAF265 | CHIR-265 | Apoptosis , Raf , VEGFR , Autophagy |
RAF265 (CHIR-265) (CHIR-265) is a potent selective inhibitor of C-Raf/B-Raf/B-Raf V600E with IC50 of 3-60 nM, and exhibits potent inhibition on VEGFR2 phosphorylation with EC50 of 30 nM. Phase 2. | |||
T40421 | 4,5-Dichlorocatechol | Others | |
4,5-Dichlorocatechol serves as a substrate for the broad-spectrum chlorocatechol 1,2-dioxygenase in Pseudomonas chlororaphis RW71. Its inhibition constant (Ki) values for the dioxygenase enzyme are 30 nM with the Chlorob... | |||
T35348 | LDN-193189 2HCl | LDN-193189 2HCl,DM-3189 2HCl | ALK , TGF-beta/Smad |
LDN-193189 2HCl (DM-3189 2HCl) is a selective BMP signaling inhibitor that inhibits ALK1,ALK2,ALK3 and ALK6, showing IC50s of 0.8 nM, 0.8 nM, 5.3 nM, and 16.7 nM, respectively, in kinase assays.LDN-193189 2HCl inhibited ... | |||
T13058 | T025 | CDK | |
T025 is a pan CLK inhibitor with Kds of 4.8, 0.096, 6.5, 0.61, and 0.074 nM for CLK1-4, respectively. T025 displays anti-proliferative activities with IC50s of 30-300 nM in hematological and solid cancer cell lines. T025... | |||
T3588 | JK184 | Hedgehog/Smoothened | |
JK184 is a potent Hedgehog (Hh) pathway inhibitor. | |||
T6143 | PI-103 | PI103,PI 103 | Apoptosis , DNA-PK , PI3K , mTOR , Autophagy |
PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK). | |||
T2610L | BMS-599626 2HCL(714971-09-2 Free base) | BMS 599626 dihydrochloride,BMS-599626 2HCL(714971-09-2 Free base),AC480 2HCl | HER |
BMS-599626 2HCL (AC480 2HCl) is a BMS-599626 derivative. BMS-599626 is an orally available and selective dual inhibitor of HER1 and HER2 with IC50s of 20 and 30 nM, respectively. BMS-599626 inhibits tumor cell proliferat... | |||
T3528 | Senicapoc | ICA-17043 | Potassium Channel |
Senicapoc (ICA-17043) is a potent inhibitor of the Gardos channel and ameliorates RBC dehydration in the SAD mouse. Senicapoc blocked Ca2+-induced rubidium flux from human RBCs with an IC50 value of 11 ± 2 nM (CLT IC50 =... |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15277 | Fervenulin | Parasite | |
Fervenulin is isolated from a nematicidal actinomycete Streptomyces sp. CMU-MH021 with nematicidal activity. It also inhibits egg hatch and J2 mortality of M. incognita (MICs: 30 μg/mL and 120 μg/mL, respectively). | |||
T13108 | Pamufetinib | H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115 | VEGFR , c-Met/HGFR |
Pamufetinib (TAS-115) is a potent inhibitor of VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase(IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively). | |||
T16791 | Rottlerin | Mallotoxin,NSC 56346,NSC 94525 | CaMK , Apoptosis , Others , HIV Protease , PKA , PKC , Autophagy |
Rottlerin (NSC-56346) is a natural product purified from Mallotus Philippinensis and is a specific PKC inhibitor (IC50: PKCδ of 3-6 μM, PKCα,β,γ of 30-42 μM, PKCε,η,ζ of 80-100 μM). Rottlerin causes apoptosis via caspase... | |||
TN1567 | Delphinidin chloride | Estrogen Receptor/ERR , VEGFR | |
Delphinidin chloride, a natural plant pigment found in berries and red wine, is a precursor of certain anthocyanins. Delphinidin chloride induces the release of nitric oxide from the vascular endothelium, resulting in va... | |||
T6717 | Vanillin | Lioxin,m-Methoxy-p-hydroxybenzaldehyde,Zimco,p-Vanillin,p-Hydroxy-m-methoxybenzaldehyde,FEMA 3107 | Others , Endogenous Metabolite |
Vanillin (Zimco) is a single molecule extracted from vanilla beans and also a popular odor used widely in perfume, food and medicine.Vanillin can reversibly and non-competitively inhibit the cellulase activity at appropr... | |||
T1411 | Terbinafine hydrochloride | KWD 2019,Terbinafine HCl,TDT 067 hydrochloride | Antibacterial , Antibiotic , Antifungal |
Terbinafine hydrochloride (KWD 2019) is a synthetic allylamine derivative structurally related to naftifine. Terbinafine is active against dermatophytes. | |||
T6702 | Terbinafine | Terbinex,SF 86-327,Lamisil,TDT 067 | Antibacterial , Antibiotic , Antifungal |
Terbinafine (TDT 067) is a synthetic allylamine derivative with antifungal activity. Terbinafine exerts its effect through inhibition of squalene epoxidase, thereby blocking the biosynthesis of ergosterol, an important c... | |||
T5S2017 | Ingenol | (-)-Ingenol | PKC |
1. Ingenol ((-)-Ingenol) mebutate is an effective treatment for actinic keratosis. 2. Formulating novel derivatives from Ingenol esters may be an innovative approach to develop new lead compounds to reactivate latent HIV... | |||
T0185 | Escitalopram | Seroplex,S-(+)-Citalopram,(S)-Citalopram | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Adrenergic Receptor , AChR , Norepinephrine , Histamine Receptor |
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol uptake in alcoholics and is used in depressed patien... | |||
T3158 | Harmane | Loturine,Harman,Aribine | Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor |
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke. | |||
TN5959 | 30-Oxopseudotaraxasterol | 3β-Hydroxytaraxaster-20-en-30-al | |
30-Oxopseudotaraxasterol is a natural product from Pulicaria canariensis ssp. lanata. | |||
TN2985 | 30-Oxolupeol | Others | |
30-Oxolupeol is a natural product of Ilex, Aquifoliaceae. The catalog number is TN2985 and the CAS number is 64181-07-3. 30-Oxolupeol can be used as a reference standard. | |||
T73561 | NK007 | ||
NK007 is a novel anti-SARS-CoV-2 agent with an EC 50 value of 30 nM. | |||
TN4835 | Przewalskin | HIV Protease | |
Przewalskin A and Przewalskin B showed modest anti-HIV-1 activity with EC50 = 41 and 30 microg/mL, respectively. | |||
TN2984 | 30-Hydroxylup-20(29)-en-3-one | Others | |
30-Hydroxylup-20(29)-en-3-one is a natural product of Maytenus, Celastraceae. The catalog number is TN2984 and the CAS number is 72944-06-0. 30-Hydroxylup-20(29)-en-3-one can be used as a reference standard. | |||
TN6135 | Methoxyimbricatin | ||
Methoxyimbricatin is a natural product for research related to life sciences. The catalog number is TN6135 and the CAS number is 233759-30-3. | |||
TN2651 | 16alpha-Hydroxybauerenol | Others | |
16alpha-Hydroxybauerenol is a natural product for research related to life sciences. The catalog number is TN2651 and the CAS number is 214351-30-1. | |||
TN6560 | Quercetin-3'-glucoside | ||
Quercetin-3'-glucoside is a natural product for research related to life sciences. The catalog number is TN6560 and the CAS number is 19254-30-9. | |||
TN2780 | 2''-O-acetyl-platyconic acid A | Others | |
2''-O-acetyl-platyconic acid A is a natural product for research related to life sciences. The catalog number is TN2780 and the CAS number is 1256935-30-4. | |||
T8204 | Gummiferin | Others | |
Gummiferin is a natural product for research related to life sciences. The catalog number is T8204 and the CAS number is 33286-30-5. | |||
TN4068 | Florosenine | Others | |
Florosenine is a natural product of Senecio, Asteraceae. The catalog number is TN4068 and the CAS number is 16958-30-8. Florosenine can be used as a reference standard. | |||
TN1380 | Marmesinin | Ammijin | Others |
Marmesinin is a natural product of Ammi, Apiaceae. The catalog number is TN1380 and the CAS number is 495-30-7. Marmesinin can be used as a reference standard. | |||
TN5768 | Chiricanine A | ||
Chiricanine A is a natural product for research related to life sciences. The catalog number is TN5768 and the CAS number is 350593-30-5. | |||
TN5377 | Nardoeudesmol A | ||
Nardoeudesmol A is a natural product for research related to life sciences. The catalog number is TN5377 and the CAS number is 1445952-30-6. | |||
TN5328 | Carabrolactone A | ||
Carabrolactone A is a natural product of Carpesium, Asteraceae. The catalog number is TN5328 and the CAS number is 1187925-30-9. Carabrolactone A can be used as a reference standard. | |||
TN3569 | Calyciphylline A | Others | |
Calyciphylline A is a natural product of Daphniphyllum, Daphniphyllaceae. The catalog number is TN3569 and the CAS number is 596799-30-3. Calyciphylline A can be used as a reference standard. | |||
TN5525 | Orientin 2''-O-rhamnoside | 2''-O-Rhamnosylorientin,Luteolin 8-C-neohesperidoside | |
Orientin 2''-O-rhamnoside is a natural product for research related to life sciences. The catalog number is TN5525 and the CAS number is 81398-30-3. | |||
TN2864 | 3',4',5',3,5,6,7-Heptamethoxyflavone | Antifection | |
3',4',5',3,5,6,7-Heptamethoxyflavone is a natural product for research related to life sciences. The catalog number is TN2864 and the CAS number is 17245-30-6. | |||
TN3661 | Cinnamyl coumarate | Others | |
Cinnamyl coumarate is a natural product for research related to life sciences. The catalog number is TN3661 and the CAS number is 115610-30-5. | |||
TN3722 | Cryptomeridiol 11-rhamnoside | Others | |
Cryptomeridiol 11-rhamnoside is a natural product for research related to life sciences. The catalog number is TN3722 and the CAS number is 349112-30-7. | |||
TN2710 | 2,4,6-Trihydroxybenzoic acid | Others | |
2,4,6-Trihydroxybenzoic acid is a natural product for research related to life sciences. The catalog number is TN2710 and the CAS number is 83-30-7. | |||
TN1748 | Humantenirine | P450 | |
Humantenirine is a natural product of Gelsemium, Loganiaceae. The catalog number is TN1748 and the CAS number is 82375-30-2. Humantenirine can be used as a reference standard. | |||
TN6086 | Machigline | ||
Machigline is a natural product for research related to life sciences. The catalog number is TN6086 and the CAS number is 87264-30-0. | |||
TN5615 | Ent-13,16β,17-Trihydroxykauran-19-oic acid | ||
ent-13,16β,17-Trihydroxykauran-19-oic acid is a natural product for research related to life sciences. The catalog number is TN5615 and the CAS number is 142543-30-4. | |||
TN2589 | 11alpha,12alpha-Epoxy-3beta,23-dihydroxy-30-norolean-20(29)-en-28,13beta-olide | Others | |
11alpha,12alpha-Epoxy-3beta,23-dihydroxy-30-norolean-20(29)-en-28,13beta-olide is a natural product from Paeonia lactiflora. | |||
TN3275 | 8-Epicrepiside E | Others | |
8-Epicrepiside E is a natural product of Saussurea, Asteraceae. The catalog number is TN3275 and the CAS number is 93395-30-3. 8-Epicrepiside E can be used as a reference standard. | |||
TN2105 | Proscillaridin A | Topoisomerase | |
Proscillaridin A is a natural product.It is a potent poison of topoisomerase I/II activity with IC50 values of 30 nM and 100 nM, respectively. | |||
T37358 | Myristelaidic Acid | ||
Myristelaidic Acid is a natural product for research related to life sciences. The catalog number is T37358 and the CAS number is 50286-30-1. | |||
TN6388 | Methyl epi-dihydrophaseate | ||
Methyl epi-dihydrophaseate is a natural product for research related to life sciences. The catalog number is TN6388 and the CAS number is 57761-30-5. | |||
TN2642 | 16,17-Dihydroapovincamine | Others | |
16,17-Dihydroapovincamine is a natural product for research related to life sciences. The catalog number is TN2642 and the CAS number is 57130-30-0. | |||
TN5994 | Elatoside E | ||
Elatoside E is a natural product for research related to life sciences. The catalog number is TN5994 and the CAS number is 156980-30-2. | |||
TN4945 | Saprirearine | Others | |
Saprirearine is a natural product of Salvia, Lamiaceae. The catalog number is TN4945 and the CAS number is 453518-30-4. Saprirearine can be used as a reference standard. | |||
TN4940 | Sanggenol P | Others | |
Sanggenol P is a natural product of Morus, Moraceae. The catalog number is TN4940 and the CAS number is 1351931-30-0. Sanggenol P can be used as a reference standard. | |||
TN5984 | 2α,3α,24-Trihydroxyursa-12,20(30)-dien-28-oic acid | ||
2α,3α,24-Trihydroxyursa-12,20(30)-dien-28-oic acid is a natural product for research related to life sciences. The catalog number is TN5984 and the CAS number is 341503-22-8. | |||
TN6357 | 5-Hydroxy-1,7-diphenylhept-6-en-3-one | ||
5-Hydroxy-1,7-diphenylhept-6-en-3-one is a natural product for research related to life sciences. The catalog number is TN6357 and the CAS number is 155239-30-8. | |||
TN6033 | Griffithazanone A | ||
Griffithazanone A is a natural product of Goniothalamus, Annonaceae. The catalog number is TN6033 and the CAS number is 240122-30-9. Griffithazanone A can be used as a reference standard. | |||
TN4766 | Phloracetophenone 4'-O-glucoside | Others | |
Phloracetophenone 4'-O-glucoside is a natural product for research related to life sciences. The catalog number is TN4766 and the CAS number is 5027-30-5. | |||
TN5893 | Toddalolactone 3′-O-ethyl ether | ||
Toddalolactone 3′-O-ethyl ether is a natural product for research related to life sciences. The catalog number is TN5893 and the CAS number is 1538607-30-5. | |||
TN5479 | Afzelechin-(4α→8)-epiafzelechin | ||
Afzelechin-(4α→8)-epiafzelechin is a natural product for research related to life sciences. The catalog number is TN5479 and the CAS number is 1383627-30-2. | |||
TN5809 | 1,4:3,6-Dianhydro-α-D-glucopyranose | ||
1,4:3,6-Dianhydro-α-D-glucopyranose is a natural product for research related to life sciences. The catalog number is TN5809 and the CAS number is 4451-30-3. | |||
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Cat No. | Product Name | Species | Expression System |
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TMPK-01116 | A30 Protein, Monkeypox virus, Recombinant (His) | Monkeypox virus | HEK293 Cells |
Monkeypox virus (MPXV) is double-stranded DNA virus belonging to the genus orthopoxvirus that causes a smallpox-like disease in humans. A30L is an envelope protein required for the fusion of virus and host cell to form s... | |||
TMPY-05051 | Influenza A H6N1 (A/quail/Hong Kong/1721-30/99) Hemagglutinin/HA1 Protein (His) | H6N1 | HEK293 Cells |
Influenza A H6N1 (A/quail/Hong Kong/1721-30/99) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.6 kDa and the accession number is Q8UWT7. | |||
TMPY-00363 | Bikunin/AMBP Protein, Human, Recombinant (aa 206-348, His) | Human | P. pastoris (Yeast) |
Bikunin/AMBP Protein, Human, Recombinant (aa 206-348, His) is expressed in yeast with His tag. The predicted molecular weight is 17.4 kDa and the accession number is CAA38587.1. | |||
TMPY-00326 | Bikunin/AMBP Protein, Human, Recombinant (mFc) | Human | HEK293 Cells |
Bikunin/AMBP Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 47.2 kDa and the accession number is P02760. | |||
TMPJ-00234 | AMBP Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Protein AMBP belongs to the calycin superfamily and Lipocalin family. AMBP can be cleaved into three chains: α-1-microglobulin, inter-α-trypsin inhibitor light chain and trypstatin. AMBP is expressed by the liver and sec... | |||
TMPY-03044 | Bikunin/AMBP Protein, Human, Recombinant (aa 1-203, His) | Human | HEK293 Cells |
Bikunin/AMBP Protein, Human, Recombinant (aa 1-203, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 22.3 kDa and the accession number is P02760. | |||
TMPK-00831 | Galectin-3 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Galectin-3 (Gal-3) is a 30 kDa β-galactose, highly conserved and widely distributed intracellularly and extracellularly. Gal-3 has been demonstrated in recent years to be a novel inflammatory factor participating in the ... | |||
TMPJ-01210 | IL-33 Protein, Mouse, Recombinant | Mouse | E. coli |
Mouse Interleukin 33 (IL-33) is a 30 kDa proinflammatory cytokine which may also regulates gene transcription in producer cells. IL-33 is constitutively expressed in smooth muscle and airway epithelia. IL-33 was identifi... | |||
TMPJ-00375 | HGF Protein, Human, Recombinant (His) | Human | HEK293 Cells |
HGF, is a pleiotropic protein in the Plasminogen subfamily of S1 peptidases and contains 4 kringle domains, 1 PAN domain and 1 peptidase S1 domain. HGF is secreted as an inactive 728 amino acid (aa) single chain propepti... | |||
TMPY-02957 | DYDC2 Protein, Human, Recombinant (GST) | Human | E. coli |
DPY30 domain containing 2 belongs to the dpy-30 family. Dumpy-30 family members act as determinants of male fertility and interaction partners of metal-responsive transcription factor 1 (MTF-1) in Drosophila. MTF-1 plays... | |||
TMPY-00496 | Influenza A H1N1 (A/Brevig Mission/1/1918) Matrix protein 1/M1 Protein (His) | H1N1 | E. coli |
Influenza A H1N1 (A/Brevig Mission/1/1918) Matrix protein 1/M1 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 30 kDa and the accession number is Q8BAC3.1. | |||
TMPY-00498 | Influenza A H3N2 (A/Aichi/2/1968) Matrix protein 1/M1 Protein (His) | H3N2 | E. coli |
Influenza A H3N2 (A/Aichi/2/1968) Matrix protein 1/M1 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 30 kDa and the accession number is I6SGW5. | |||
TMPH-03722 | Coagulase/fibrinolysin Protein, Yersinia pestis, Recombinant (His & Myc) | Yersinia pestis | E. coli |
Seems to play an essential role in plague transmission by mediating flea blockage in a temperature-dependent fashion. Fibrinolytic activity prevails at 37 degrees Celsius whereas coagulase expression predominates at lowe... | |||
TMPK-01183 | CDCP1 Protein, Human, Recombinant (aa 30-368, His) | Human | HEK293 Cells |
Tumor metastasis depends on the dynamic regulation of cell adhesion through β1-integrin. The Cub-Domain Containing Protein-1, CDCP1, is a transmembrane glycoprotein which regulates cell adhesion. Overexpression and loss ... | |||
TMPJ-01054 | PAFAHB Protein, Human, Recombinant (His) | Human | E. coli |
Platelet-Activating Factor Acetylhydrolase IB Subunit β (PAFAHB) is a cytoplasmic hydrolase. PAFAHB is a member of the GDSL lipolytic enzyme family. It also belongs to Platelet-activating factor acetylhydrolase IB beta/g... | |||
TMPK-00336 | GPC3 Protein-VLP, Human, Recombinant | Human | E. coli |
Glypican-3 is a protein ,which is encoded by the GPC3 gene in humans.The protein core of GPC3 consists of two subunits, where the N-terminal subunit has a size of ~40 kDa and the C-terminal subunit is ~30 kDa.Glypican 3 ... | |||
TMPK-00337 | GPC3 Protein-VLP, Human, Recombinant (aa 438-554) | Human | HEK293 Cells |
Glypican-3 is a protein ,which is encoded by the GPC3 gene in humans.The protein core of GPC3 consists of two subunits, where the N-terminal subunit has a size of ~40 kDa and the C-terminal subunit is ~30 kDa.Glypican 3 ... | |||
TMPJ-01449 | 3CLpro/3C-like Protease Protein, SARS-CoV-2, Recombinant | SARS-CoV-2 | E. coli |
The viral main proteinase (M pro , also called 3CL pro ), which controls the activities of the coronavirus replication complex. It functions as a cysteine protease engaging in the proteolytic cleavage of the viral precur... | |||
TMPH-02046 | Ribonuclease 7 Protein, Human, Recombinant (His) | Human | E. coli |
Exhibits a potent RNase activity. Has broad-spectrum antimicrobial activity against many pathogenic microorganisms and remarkably potent activity (lethal dose of 90% < 30 nM) against a vancomycin resistant Enterococcus f... | |||
TMPK-00351 | RANK/TNFRSF11A Protein, Human, Recombinant (aa 30-212, hFc) | Human | HEK293 Cells |
TNFRSF11A, also known as receptor activator of NF-κB (RANK), activates several signaling pathways, such as NF-κB, JNK, ERK, p38α, and Akt/PKB. RANK/TNFRSF11A is a novel and frequent target for de novo methylation in glio... | |||
TMPY-03268 | GABARAPL1 Protein, Human, Recombinant (His) | Human | E. coli |
ATG8, also known as GABARAPL1, is a ubiquitin-like protein that has a crystal structure. ATG8 consists of a 5-stranded β-sheet, which is enclosed by two α-helices at one side and one α-helix at the other side and exhibit... | |||
TMPJ-01390 | MINPP1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Multiple Inositol Polyphosphate Phosphatase 1/MINPP1 is an enzyme that removes 3-phosphate from inositol phosphate substrates. MINPP1 also converts 2,3 bisphosphoglycerate (2,3-BPG) to 2-phosphoglycerate. MINPP1 is synth... | |||
TMPK-00062 | CD160 Protein, Human, Recombinant (His & Avi) | Human | HEK293 Cells |
CD160 (also Natural killer cell receptor BY55) is a 27 ‑ 30 kDa member of the Ig superfamily. In human, it is expressed principally on nonmyeloid hematopoietic cells. CD160 antigenis a receptor on immune cells capable to... | |||
TMPJ-01371 | Limitin Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Limitin, also called IFN-ζ, is a secreted interferon (IFN)-like glycoprotein. Limitin has approximately 30% sequence homology with IFN-α, IFN-β, and IFN-ω and binds to the IFN-α/β receptors. Like IFN-α and IFN-β, limitin... | |||
TMPJ-00075 | CD27 Ligand/CD70 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
CD27 Ligand (CD70) is a 30 kDa type 2 transmembrane glycoproteinis that belongs to the tumor necrosis factor (TNF) ligand family.Human CD27 Ligand extracellular region is 64% aa identical to mouse and rat CD27 Ligand ext... | |||
TMPY-03288 | USP30 Protein, Human, Recombinant (SUMO) | Human | Baculovirus Insect Cells |
Ubiquitin specific peptidase 30, also known as USP30, is a deubiquitinating enzyme that is embedded in the mitochondrial outer membrane. Depletion of USP30 expression by RNA interference induced elongated and interconnec... | |||
TMPJ-00018 | CCL16 Protein, Human, Recombinant | Human | E. coli |
CCL16 is a member of CC chemokine family. CCL16 cDNA encodes a 120 amino acid peptide along with a 23 amino acids signal peptide that is cleaved to generate 97 amino acid protein. CCL16 is distantly related to other CC c... | |||
TMPJ-00674 | RANK/TNFRSF11A Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Receptor activator of NF-κB(RANK,TNFRSF11A) belongs to one member of tumor necrosis factor receptor family.It is a receptor for TNFSF11/RANKL/TRANCE/OPGL. This gene encodes a type 1 membrane protein with a 30 amino acid... | |||
TMPJ-00667 | DEFB4A Protein, Human, Recombinant | Human | E. coli |
β-Defensin 4A is a membrane-active cationic peptide that functions in inflammation and innate immune responses. There are at least 30 β-Defensins, which are distinguished from α-Defensins by the connectivity pattern of t... | |||
TMPJ-00873 | CCL3L1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
C-C Motif Chemokine 3-Like 1 (CCL3L1) is a secreted protein that belongs to the intercrine beta (chemokine CC) family. CCL3L1 is a ligand for CCR1, CCR3 and CCR5. CCL3L1 binds to several chemokine receptors including che... | |||
TMPY-02599 | MDH1 Protein, Rat, Recombinant (His) | Rat | E. coli |
Malate dehydrogenases 1(MDH1 / MDHA) is a soluble form of malate dehydrogenases. Malate dehydrogenases (MDH) is a group of multimeric enzymes consisting of identical subunits usually organized as either dimer or tetramer... | |||
TMPJ-01425 | SARS-CoV-2 NSP1 Protein (His) | SARS-CoV-2 | E. coli |
The Severe Acute Respiratory Syndrome (SARS) Coronavirus (CoV) is an enveloped, positive-stranded RNA viruses that can cause a severe respiratory disease. Its genome consists of a ∼30 kb linear, non-segmented, capped, po... | |||
TMPH-02349 | Influenza A H1N1 (strain A/Malaysia:Malaya/302/1954) Non-structural protein 1 (His & Myc) | H1N1 | E. coli |
Prevents the establishment of the cellular antiviral state by inhibiting TRIM25-mediated DDX58 ubiquitination, which normally triggers the antiviral transduction signal that leads to the activation of type I IFN genes by... | |||
TMPK-01422 | Peptide Ready HLA-A*02:01&B2M Monomer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Peptide Ready HLA-A*02:01&B2M Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-A*02:01. Peptide ready MHC molecules comprising human HLA alleles and B2M,... | |||
TMPK-01415 | APC-equivalent Peptide Ready HLA-A*02:01&B2M Tetramer Protein, Human, MHC (His) | Human | HEK293 Cells |
Peptide Ready HLA-A*02:01&B2M Tetramer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-A*02:01. Peptide ready MHC molecules comprising human HLA alleles and B2M... | |||
TMPK-01421 | Peptide Ready HLA-A*02:01&B2M Monomer Protein, Human, MHC (His & Avi), Biotinylated | Human | HEK293 Cells |
HLA-A*02:01&B2M&Peptide ready Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-A*02:01. Peptide ready MHC molecules comprising human HLA alleles and B2M,... | |||
TMPK-01419 | Peptide Ready HLA-A*03:01&B2M Monomer Protein, Human, MHC (His & Avi), Biotinylated | Human | HEK293 Cells |
Peptide Ready HLA-A*03:01&B2M Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-A*03:01. Peptide ready MHC molecules comprising human HLA alleles and B2M,... | |||
TMPK-01425 | Peptide Ready HLA-A*11:01&B2M Monomer Protein, Human, MHC (His & Avi), Biotinylated | Human | HEK293 Cells |
Peptide Ready HLA-A*11:01&B2M Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-A*11:01. Peptide ready MHC molecules comprising human HLA alleles and B2M,... | |||
TMPK-01426 | Peptide Ready HLA-A*11:01&B2M Monomer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Peptide Ready HLA-A*11:01&B2M Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-A*11:01. Peptide ready MHC molecules comprising human HLA alleles and B2M,... | |||
TMPK-01409 | Peptide Ready HLA-A*24:02&B2M Monomer Protein, Human, MHC (His & Avi), Biotinylated | Human | HEK293 Cells |
Peptide Ready HLA-G&B2M Monomer is absent from peptide, namely peptide-receptive MHC. It can be loaded with antigenic peptides matching HLA-G. Peptide ready MHC molecules comprising human HLA alleles and B2M, which can b... | |||
TMPK-01455 | HLA-A*02:01&B2M&PRAME (SLLQHLIGL) Monomer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
PRAME (PReferentially expressed Antigen in MElanoma) is a melanoma-associated antigen expressed in cutaneous and ocular melanomas and some other malignant neoplasms, while its expression in normal tissue and benign tumor... | |||
TMPK-01406 | HLA-A*02:01&B2M&PRAME (SLLQHLIGL) Tetramer Protein, Human, MHC (His & Avi), PE-Labeled | Human | HEK293 Cells |
PRAME (PReferentially expressed Antigen in MElanoma) is a melanoma-associated antigen expressed in cutaneous and ocular melanomas and some other malignant neoplasms, while its expression in normal tissue and benign tumor... | |||
TMPK-01432 | HLA-A*11:01&B2M&KRAS G12A (VVVGAAGVGK) Tetramer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Kirsten rat sarcoma 2 viral oncogene homolog (KRAS) is the most commonly mutated oncogene in human cancer. The developments of many cancers depend on sustained expression and signaling of KRAS, which makes KRAS a high-pr... | |||
TMPK-01445 | HLA-A*02:01&B2M&MAGE-A1 (KVLEYVIKV) Monomer Protein, Human, MHC (His & Avi), Biotinylated | Human | HEK293 Cells |
MAGE-A1 belongs to the chromosome X-clustered genes of cancer-testis antigen family and is normally expressed in the human germ line but is also overexpressed in various tumors. | |||
TMPK-01468 | HLA-A*02:01&B2M&MART-1 (ELAGIGILTV) Tetramer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Melanoma antigen recognized by T cell-1 (Mart-1), one of the melanosome-specific proteins, also recognized by cytotoxicity T lymphocytes as a marker. Mart-1 is considered to play a critical role in the immunotherapy for ... | |||
TMPK-01459 | HLA-A*02:01&B2M&MAGE-A4 or MAGE-A8 (KVLEHVVRV) Monomer Protein, Human, MHC (His & Avi), Biotinylated | Human | HEK293 Cells |
MAGE-A4 and MAGE-A8 are type I membes of the melanoma associated antigen (MAGE) family. The MAGE family is a large, highly conserved group of proteins that share a common MAGE homology domain. Both MAGE-A4 and MAGE-A8 an... | |||
TMPK-01495 | HLA-A*01:01&B2M&MAGE-A3 (EVDPIGHLY) Monomer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Melanoma antigen gene A3 (MAGE-A3) is one of the most immunogenic cancer testis antigens and is common in various types of cancers. MAGE-A3 can be considered as a predictor for poor prognosis and an option for vaccine im... | |||
TMPK-01433 | HLA-A*11:01&B2M&KRAS G12C (VVVGACGVGK) Tetramer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Kirsten rat sarcoma 2 viral oncogene homolog (KRAS) is the most commonly mutated oncogene in human cancer. The developments of many cancers depend on sustained expression and signaling of KRAS, which makes KRAS a high-pr... | |||
TMPK-01482 | HLA-A*02:03&B2M&AFP (FMNKFIYEI) Tetramer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Alpha-fetoprotein (AFP), a specific liver cancer marker, T cells expressing AFP-CAR selectively degranulated, released cytokines, and lysed liver cancer cells that were HLA-A*02:01 /AFP while sparing cells from multiple ... | |||
TMPK-01496 | HLA-A*01:01&B2M&CT83 (NTDNNLAVY) Monomer Protein, Human, MHC (His & Avi) | Human | HEK293 Cells |
Cancer/testis antigens 83 (CT83), also called KK-LC-1 or CXorf61, recognized by cytotoxic T lymphocytes (CTL), has become a promising target for immunotherapy. | |||
------------------------ More ------------------------ |
Cat No. | Product Name | ||
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L8800 | Drug-Fragment Library | 1119 compounds | |
1119 drug fragments,a must-have tool for FBDD; | |||
L2520 | Glycometabolism Compound Library | 702 compounds | |
702 glycometabolism-related comounds, can be used for HTS and HCT; | |||
L6130 | Terpene Natural Product Library | 516 compounds | |
A unique collection of 516 natural terpenes and terpenoids can be used for high throughput and high content screening; | |||
L5700 | Featured Fragment Library | 246 compounds | |
A unique collection of 246 fragment-like small molecules for FBDD; | |||
L2190 | Anti-Lung Cancer Compound Library | 1702 compounds | |
A unique collection of 1702 compounds with anti-lung cancer therapeutic activity or targeting lung cancer’s major signaling pathways, can be used for anti-lung cancer drug discovery and mechanism study; |